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Synthesis of Vixotrigine, a Use-Dependent Sodium Channel Blocker. Part 1: Development of Bulk Supply Routes to Enable Proof of Concept

Authors :
Michael Williams
William F. Kiesman
Gerard M. P. Giblin
Adrian Heseltine
David T. MacPherson
James A. Ramsden
Ravi Vadali
David R Witty
Source :
Organic Process Research & Development. 24:2802-2813
Publication Year :
2020
Publisher :
American Chemical Society (ACS), 2020.

Abstract

Two syntheses of vixotrigine are reported. Route 1, adapted from the medicinal chemistry route, enabled rapid delivery of drug substance for clinical development. Route 2, which was developed to ad...

Details

ISSN :
1520586X and 10836160
Volume :
24
Database :
OpenAIRE
Journal :
Organic Process Research & Development
Accession number :
edsair.doi...........b6912304c8c05f1fa22e5aed2df15343
Full Text :
https://doi.org/10.1021/acs.oprd.0c00382