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Inhibition of guinea pig aldehyde oxidase activity by different flavonoid compounds: An in vitro study
- Source :
- Bioorganic chemistry. 64
- Publication Year :
- 2015
-
Abstract
- Aldehyde oxidase (AO), a cytosolic molybdenum-containing hydroxylase, is predominantly active in liver and other tissues of mammalian species and involved in the metabolism of extensive range of aldehydes and nitrogen-containing compounds. A wide range of natural components including polyphenols are able to interfere with AO-catalyzed reactions. Polyphenols and flavonoids are one of the extensive secondary plant metabolites ubiquitously present in plants considered an important part of the human diet. The aim of the present study was to investigate inhibitory effect of selected phenolic compounds from three subclasses of aurone, flavanone and phenolic lactone compounds on the activity of AO, spectrophotometrically. AO enzyme was partially purified from liver of guinea pig. Then, inhibitory effects of 10 flavonoid compounds including 8 derivatives of 2-benzylidenebenzofuran-3(2H)-ones, as well as naringenin and ellagic acid on the activity of aldehyde oxidase were assessed compared with the specific inhibitor of AO, menadione. Among the phenolic compounds with inhibitory effects on the enzyme, ellagic acid (IC50=14.47 μM) was the most potent agent with higher inhibitory action than menadione (IC50=31.84 μM). The mechanisms by which flavonoid compounds inhibit AO activity have been also determined. The inhibitory process of the assessed compounds occurs via either a non-competitive or mixed mode. Although flavonoid compounds extensively present in the nature, mainly in dietary regimen, aurones with promising biological properties are not widely distributed in nature, so synthesis of aurone derivatives is of great importance. Additionally, aurones seem to provide a promising scaffold in medicinal chemistry for the skeleton of new developing drugs, so the results of the current study can be valuable in order to better understanding drug-food as well as drug-drug interaction and also appears to be worthwhile in drug development strategies.
- Subjects :
- 0301 basic medicine
Naringenin
Male
Flavonoid
Guinea Pigs
Ligands
Biochemistry
Benzylidene Compounds
03 medical and health sciences
chemistry.chemical_compound
0302 clinical medicine
Menadione
Ellagic Acid
Drug Discovery
Aurone
Animals
Enzyme Inhibitors
Molecular Biology
Aldehyde oxidase
Benzofurans
Enzyme Assays
chemistry.chemical_classification
Flavonoids
Organic Chemistry
food and beverages
Aldehyde Oxidase
Molecular Docking Simulation
Kinetics
030104 developmental biology
chemistry
Liver
Polyphenol
030220 oncology & carcinogenesis
Flavanone
Ellagic acid
Subjects
Details
- ISSN :
- 10902120
- Volume :
- 64
- Database :
- OpenAIRE
- Journal :
- Bioorganic chemistry
- Accession number :
- edsair.doi.dedup.....096acaa9dee16abe93776bed9e2d1c34