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A New Method for Chemoselective Conjugation of Unprotected Peptides to Dauno- and Doxorubicin

Authors :
Marina Taliani
Antonello Pessi
Daniela Fattori
Annalise Di Marco
Paolo Ingallinella
Source :
Bioorganic & Medicinal Chemistry Letters. 11:1343-1346
Publication Year :
2001
Publisher :
Elsevier BV, 2001.

Abstract

A new approach for chemoselective ligation of peptides to dauno- and doxorubicin through an oxime bond is presented. The method does not require protecting groups on the peptide moiety.

Details

ISSN :
0960894X
Volume :
11
Database :
OpenAIRE
Journal :
Bioorganic & Medicinal Chemistry Letters
Accession number :
edsair.doi.dedup.....4022d423d209963354d4ec1fd096d378
Full Text :
https://doi.org/10.1016/s0960-894x(01)00223-2