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2-Aryloxymethylmorpholine histamine H(3) antagonists

Authors :
Kirsten L. Miller
Michael A. Letavic
Diane Nepomuceno
Pascal Bonaventure
Brian Lord
Kiev S. Ly
John M. Keith
Nicholas I. Carruthers
S. Timothy Motley
Steven W. Sutton
Mark A. Feinstein
Source :
Bioorganicmedicinal chemistry letters. 18(21)
Publication Year :
2008

Abstract

The synthesis and biological activity of a new series of 2-aryloxymethylmorpholine histamine H 3 antagonists is described. The new compounds are high affinity histamine H 3 ligands that penetrate the CNS and occupy the histamine H 3 receptor in rat brain.

Details

ISSN :
14643405
Volume :
18
Issue :
21
Database :
OpenAIRE
Journal :
Bioorganicmedicinal chemistry letters
Accession number :
edsair.doi.dedup.....5bd19ccd5a4b70ad5040aaa25493538d