1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure–affinity relationships and molecular modeling studies

Authors :: Daniela Catarzi
Flavia Varano
Daniela Poli
Lucia Squarcialupi
Marco Betti
Letizia Trincavelli
Claudia Martini
Diego Dal Ben
Ajiroghene Thomas
Rosaria Volpini
Vittoria Colotta
Source :: Università degli studi di Firenze-IRIS
Publication Year :: 2015
Publisher :: Elsevier BV, 2015.

Subjects :: G protein-coupled receptors
Organic Chemistry
Clinical Biochemistry
Drug Discovery
Tricyclic heteroaromatic systems
Pharmaceutical Science
Molecular Medicine
Adenosine receptor antagonists
Triazoloquinoxalines
Ligand-receptor modeling studies
Molecular Biology
Biochemistry

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