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A Cross-Metathesis Route to Functionalized α-Methyl α-Substituted Amino Acids

Authors :
Lavinia Panella
Roy P. M. Storcken
Hans E. Schoemaker
Floris P. J. T. Rutjes
Floris L. van Delft
Quirinus B. Broxterman
Bernard Kaptein
Source :
Advanced Synthesis & Catalysis, 349, 161-164, Advanced Synthesis & Catalysis, 349, 1-2, pp. 161-164
Publication Year :
2007
Publisher :
Wiley, 2007.

Abstract

A chemoenzymatic approach to the synthesis of functionalized α-methyl α-substituted amino acids is detailed. This involves amidase-mediated enzymatic resolution of α-methyl α-substituted side-chain ω-unsaturated amino acids followed by functionalization via cross-metathesis.

Details

ISSN :
16154169 and 16154150
Volume :
349
Database :
OpenAIRE
Journal :
Advanced Synthesis & Catalysis
Accession number :
edsair.doi.dedup.....80a28359ce99a7addccee83f060c2b72
Full Text :
https://doi.org/10.1002/adsc.200600446