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One-Pot Synthesis of 2-Pyridones via Chemo- and Regioselective Tandem Blaise Reaction of Nitriles with Propiolates

Authors :
Hyunik Shin
Joo Yeon Hong
Ka Yeon Ryu
Yu Sung Chun
Jongki Hong
Sang‐gi Lee
Young Ok Ko
Source :
The Journal of Organic Chemistry. 74:7556-7558
Publication Year :
2009
Publisher :
American Chemical Society (ACS), 2009.

Abstract

The Blaise reaction intermediate, generated in situ from Reformatsky reagent and nitrile, reacted with propiolates in a chemo- and regioselective manner to afford 2-pyridone derivatives in good to excellent yields.

Details

ISSN :
15206904 and 00223263
Volume :
74
Database :
OpenAIRE
Journal :
The Journal of Organic Chemistry
Accession number :
edsair.doi.dedup.....e9a3cdbde38fbb2906a3b590c52a282c
Full Text :
https://doi.org/10.1021/jo901642t