Back to Search Start Over

Discovery of Hexahydrofuro[3,2

Authors :
Shan, Li
Hongfei, Si
Xiaojuan, Song
Chong, Lei
Xiaoqiang, He
Jie, Wang
Yiling, Liu
Yang, Zhou
Jian-Guo, Song
Lijie, Peng
Xia, Tang
Shingpan, Chan
Xiaomei, Ren
Zhengchao, Tu
Zhengqiu, Li
Zhen, Wang
Zhang, Zhang
Ke, Ding
Source :
Journal of medicinal chemistry. 65(15)
Publication Year :
2022

Abstract

Janus kinase 3 (JAK3) is a potential target for the treatment of hematological malignancies. Herein, we report the discovery of a series of new orally bioavailable irreversible JAK3 kinase inhibitors. The representative compound

Details

ISSN :
15204804
Volume :
65
Issue :
15
Database :
OpenAIRE
Journal :
Journal of medicinal chemistry
Accession number :
edsair.pmid..........78640a488f5fd8916f688e91a8b71f0b