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Activation and signaling mechanism revealed by GPR119-Gs complex structures

Authors :
Yuxia Qian
Jiening Wang
Linlin Yang
Yanru Liu
Lina Wang
Wei Liu
Yun Lin
Hong Yang
Lixin Ma
Sheng Ye
Shan Wu
Anna Qiao
Source :
Nature Communications, Vol 13, Iss 1, Pp 1-10 (2022)
Publication Year :
2022
Publisher :
Nature Portfolio, 2022.

Abstract

Agonists selectively targeting GPR119 hold promise for treating metabolic disorders. Here, authors reveal that GPR119 adopts a non-canonical consensus structural scaffold with an extended ligand-binding pocket for chemically different agonists.

Subjects

Subjects :
Science

Details

Language :
English
ISSN :
20411723
Volume :
13
Issue :
1
Database :
Directory of Open Access Journals
Journal :
Nature Communications
Publication Type :
Academic Journal
Accession number :
edsdoj.1a5e75195b15441ab9ae910d66ae194b
Document Type :
article
Full Text :
https://doi.org/10.1038/s41467-022-34696-6