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Histone Parylation factor 1 contributes to the inhibition of PARP1 by cancer drugs

Authors :
Johannes Rudolph
Genevieve Roberts
Karolin Luger
Source :
Nature Communications, Vol 12, Iss 1, Pp 1-11 (2021)
Publication Year :
2021
Publisher :
Nature Portfolio, 2021.

Abstract

PARP1 is the target of clinically approved anti-cancer drugs whose in vivo efficacy has been hard to predict. Here the authors show how an altered active site formed between PARP1 and Histone PARylation Factor 1 (HPF1) changes the efficacy of some of these inhibitors.

Subjects

Subjects :
Science

Details

Language :
English
ISSN :
20411723
Volume :
12
Issue :
1
Database :
Directory of Open Access Journals
Journal :
Nature Communications
Publication Type :
Academic Journal
Accession number :
edsdoj.33d6d10fa6924050954dfbd2aa320cee
Document Type :
article
Full Text :
https://doi.org/10.1038/s41467-021-20998-8