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Maprotiline restores ER homeostasis and rescues neurodegeneration via Histamine Receptor H1 inhibition in retinal ganglion cells

Authors :
Wei Chen
Pingting Liu
Dong Liu
Haoliang Huang
Xue Feng
Fang Fang
Liang Li
Jian Wu
Liang Liu
David E. Solow-Cordero
Yang Hu
Source :
Nature Communications, Vol 13, Iss 1, Pp 1-18 (2022)
Publication Year :
2022
Publisher :
Nature Portfolio, 2022.

Abstract

ER stress is associated with various neurodegenerative diseases. This study found that FDA approved drug, maprotiline, inhibits histamine receptor H1-mediated ER stress and provides significant neuroprotection in mouse glaucoma model.

Subjects

Subjects :
Science

Details

Language :
English
ISSN :
20411723
Volume :
13
Issue :
1
Database :
Directory of Open Access Journals
Journal :
Nature Communications
Publication Type :
Academic Journal
Accession number :
edsdoj.3ca727977d4eaab1ecad19f6b088c6
Document Type :
article
Full Text :
https://doi.org/10.1038/s41467-022-34682-y