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BRD4-mediated repression of p53 is a target for combination therapy in AML

Authors :
Anne-Louise Latif
Ashley Newcombe
Sha Li
Kathryn Gilroy
Neil A. Robertson
Xue Lei
Helen J. S. Stewart
John Cole
Maria Terradas Terradas
Loveena Rishi
Lynn McGarry
Claire McKeeve
Claire Reid
William Clark
Joana Campos
Kristina Kirschner
Andrew Davis
Jonathan Lopez
Jun-ichi Sakamaki
Jennifer P. Morton
Kevin M. Ryan
Stephen W. G. Tait
Sheela A. Abraham
Tessa Holyoake
Brian Higgins
Xu Huang
Karen Blyth
Mhairi Copland
Timothy J. T. Chevassut
Karen Keeshan
Peter D. Adams
Source :
Nature Communications, Vol 12, Iss 1, Pp 1-16 (2021)
Publication Year :
2021
Publisher :
Nature Portfolio, 2021.

Abstract

MDM2 and BET inhibitors have shown efficacy in AML treatment. Here, the authors show that the two compounds can synergize through both p53 protein stabilization and inhibition of BRD4-mediated repression of p53 target genes.

Subjects

Subjects :
Science

Details

Language :
English
ISSN :
20411723
Volume :
12
Issue :
1
Database :
Directory of Open Access Journals
Journal :
Nature Communications
Publication Type :
Academic Journal
Accession number :
edsdoj.4058dbf2924543a399c2f17c8fd2a6ad
Document Type :
article
Full Text :
https://doi.org/10.1038/s41467-020-20378-8