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Chalcone derivatives antagonize interactions between the human oncoprotein MDM2 and p53

Authors :
Stoll, Raphael
Renner, Christian
Hansen, Silke
Palme, Stefan
Klein, Christian
Belling, Anja
Zeslawski, Wojciech
Kamionka, Marius
Rehm, Till
Muhlhahn, Peter
Schumacher, Ralf
Hesse, Friederike
Kaluza, Brigitte
Voelter, Wolfgang
Engh, Richard A.
Holak, Tad A.
Source :
Biochemistry. Jan 16, 2001, Vol. 40 Issue 2, p336, 9 p.
Publication Year :
2001

Abstract

Research has been conducted on the oncoprotein MDM2 inhibiting the tumor suppressor protein p53. Results of the multidimensional NMR spectroscopy indicate that chalcones are MDM2's inhibitors binding to the p53 binding cleft substrate of human MDM2.

Details

ISSN :
00062960
Volume :
40
Issue :
2
Database :
Gale General OneFile
Journal :
Biochemistry
Publication Type :
Academic Journal
Accession number :
edsgcl.77076859