33 results on '"Spring, David R."'
Search Results
2. Site-selective peptide functionalisation mediated via vinyl-triazine linchpins
3. Peroxide-cleavable linkers for antibody–drug conjugates
4. Disulfide re-bridging reagents for single-payload antibody-drug conjugates
5. Antibody dual-functionalisation enabled through a modular divinylpyrimidine disulfide rebridging strategy
6. Divinylpyrimidine reagents generate antibody–drug conjugates with excellent in vivo efficacy and tolerability
7. Development of small cyclic peptides targeting the CK2α/β interface
8. A dual-enzyme cleavable linker for antibody–drug conjugates
9. Fsp3-rich and diverse fragments inspired by natural products as a collection to enhance fragment-based drug discovery
10. Total synthesis and biological evaluation of simplified aplyronine analogues as synthetically tractable anticancer agents
11. An efficient, stereocontrolled and versatile synthetic route to bicyclic partially saturated privileged scaffolds
12. C(sp3)–H arylation to construct all-syn cyclobutane-based heterobicyclic systems: a novel fragment collection
13. Targeted covalent inhibitors of MDM2 using electrophile-bearing stapled peptides
14. Macrocyclisation and functionalisation of unprotected peptides via divinyltriazine cysteine stapling
15. C(sp3)–H arylation to construct all-syn cyclobutane-based heterobicyclic systems: a novel fragment collection.
16. Fsp3-rich and diverse fragments inspired by natural products as a collection to enhance fragment-based drug discovery.
17. Computationally-guided optimization of small-molecule inhibitors of the Aurora A kinase–TPX2 protein–protein interaction
18. Coumarin-derived transformable fluorescent sensor for Zn2+
19. Development of off–on fluorescent probes for heavy and transition metal ions
20. A selective and ratiometric Cu2+ fluorescent probe based on naphthalimide excimer–monomer switching
21. 3D small-molecule microarrays
22. The discovery of antibacterial agents using diversity-oriented synthesis
23. Identification of an anti-MRSA dihydrofolate reductase inhibitor from a diversity-oriented synthesis
24. Exploiting domino enyne metathesis mechanisms for skeletal diversity generation
25. Fluorous tagged small molecule microarrays
26. Copper catalyzed oxidation of organozinc halides
27. Skeletal diversity construction via a branching synthetic strategy
28. Aryl–aryl coupling via directed lithiation and oxidation
29. Diversity-oriented synthesis of bicyclic and tricyclic alkaloids.
30. Towards quorum-quenching catalytic antibodies.
31. Skeletal diversity construction viaa branching synthetic strategyElectronic supplementary information (ESI) available: Full experimental details, characterization and spectra of key compounds. See DOI: 10.1039/b607710bThe HTML version of this article has been enhanced with colour images.
32. Highlights from the 39thESFEUCHEM Conference on Stereochemistry, Bürgenstock, Switzerland, April 2004
33. Aryl–aryl coupling viadirected lithiation and oxidationElectronic supplementary information ESI available: analytical and spectroscopic data for all new compounds. See http://www.rsc.org/suppdata/cc/b5/b501939g/
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