1,062 results on '"Spring, David R."'
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2. CK2 Inhibitors Targeting Inside and Outside the Catalytic Box
3. Unlocking Amides: A General Method for the Self‐Immolative Release of Amide‐Containing Molecules
4. Tuneable thiol exchange linkers for traceless drug release applications in prodrugs and ADCs.
5. Photoredox C(2)-Arylation of Indole- and Tryptophan-Containing Biomolecules.
6. Site-selective peptide functionalisation mediated via vinyl-triazine linchpins
7. Red-light modulated ortho-chloro azobenzene photoswitch for peptide stapling via aromatic substitution
8. Microscopy and chemical analyses reveal flavone-based woolly fibres extrude from micron-sized holes in glandular trichomes of Dionysia tapetodes
9. Energetics of lipid transport by the ABC transporter MsbA is lipid dependent
10. Synthesis of structurally diverse biflavonoids
11. A recombinant approach for stapled peptide discovery yields inhibitors of the RAD51 recombinase.
12. Tryptophan in Multicomponent Petasis Reactions for Peptide Stapling and Late‐Stage Functionalisation
13. Novel non-ATP competitive small molecules targeting the CK2 α/β interface
14. Hybrid Androgen Receptor Inhibitors Outperform Enzalutamide and EPI‐001 in in vitro Models of Prostate Cancer Drug Resistance
15. Finding New Components of the Target of Rapamycin (TOR) Signaling Network through Chemical Genetics and Proteome Chips
16. Selective inhibitors of the Aurora A-TPX2 protein-protein interaction exhibit in vivo efficacy as targeted anti-mitotic agents
17. A Recombinant Approach For Stapled Peptide Discovery Yields Inhibitors of the RAD51 Recombinase
18. The human proton pump inhibitors inhibit Mycobacterium tuberculosis rifampicin efflux and macrophage-induced rifampicin tolerance
19. A fragment-based approach leading to the discovery of a novel binding site and the selective CK2 inhibitor CAM4066
20. A cryptic hydrophobic pocket in the polo-box domain of the polo-like kinase PLK1 regulates substrate recognition and mitotic chromosome segregation
21. A cell-active cyclic peptide targeting the Nrf2/Keap1 protein–protein interaction.
22. Disulfide re-bridging reagents for single-payload antibody-drug conjugates.
23. Studies Towards the Synthesis of the Core of Endiandric Acid H
24. Front Cover: Hybrid Androgen Receptor Inhibitors Outperform Enzalutamide and EPI‐001 in in vitro Models of Prostate Cancer Drug Resistance (ChemMedChem 2/2023)
25. Identification of macrocyclic peptides which activate bacterial cylindrical proteases
26. Synthesis of sp3-rich heterocyclic frameworks by a divergent synthesis strategy
27. Peroxide-cleavable linkers for antibody–drug conjugates
28. A cell-active peptide targeting the Nrf2/Keap1 protein-protein interaction
29. Studies on the biomimetic synthesis of the manzamine alkaloids
30. An expedient strategy for the diversity-oriented synthesis of macrocyclic compounds with natural product-like characteristics
31. Chapter 2. The Application of Diversity-oriented Synthesis in Chemical Biology
32. Divinylpyrimidine reagents generate antibody-drug conjugates with excellent in vivo efficacy and tolerability
33. Synthesis of sp3-rich heterocyclic frameworks by a divergent synthesis strategy.
34. Divergent and concise total syntheses of dihydrochalcones and 5-deoxyflavones recently isolated from Tacca species and Mimosa diplotricha
35. Overcoming Chemical, Biological, and Computational Challenges in the Development of Inhibitors Targeting Protein-Protein Interactions
36. Studies towards the synthesis of indolizin-5(3H)-one derivatives and related 6,5-azabicyclic scaffolds by ring-closing metathesis
37. LGR5 targeting molecules as therapeutic agents for multiple cancer types
38. Multifunctional supramolecular polymer networks as next-generation consolidants for archaeological wood conservation
39. Rapid and robust cysteine bioconjugation with vinylheteroarenes
40. Antiplasmodial and trypanocidal activity of violacein and deoxyviolacein produced from synthetic operons
41. A unified in vitro to in vivo fluorescence lifetime screening platform yields amyloid β aggregation inhibitors
42. Applications of small molecule activators and inhibitors of quorum sensing in Gram-negative bacteria
43. Hybrid Androgen Receptor Inhibitors Outperform Enzalutamide and EPI‐001 in in vitro Models of Prostate Cancer Drug Resistance.
44. Non-internalising antibody–drug conjugates.
45. A two-component 'double-click' approach to peptide stapling
46. Antibody dual-functionalisation enabled through a modular divinylpyrimidine disulfide rebridging strategy
47. Divinylpyrimidine reagents generate antibody–drug conjugates with excellent in vivo efficacy and tolerability
48. All-in-one disulfide bridging enables the generation of antibody conjugates with modular cargo loading
49. Development of small cyclic peptides targeting the CK2α/β interface
50. Correction: The multifaceted nature of antimicrobial peptides: current synthetic chemistry approaches and future directions
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